Cart
sales@molnova.com
Deltorphin I(TFA)
CAS No. 122752-15-2
Deltorphin I(TFA)( Deltorphin 1 | Deltorphin C )
Catalog No. M21043 CAS No. 122752-15-2
Deltorphin I(TFA) is an agonist of δ-opioid receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 87 | In Stock |
|
| 5MG | 160 | In Stock |
|
| 10MG | 241 | In Stock |
|
| 25MG | 408 | In Stock |
|
| 50MG | 590 | In Stock |
|
| 100MG | 826 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameDeltorphin I(TFA)
-
NoteResearch use only, not for human use.
-
Brief DescriptionDeltorphin I(TFA) is an agonist of δ-opioid receptor.
-
DescriptionDeltorphin I(TFA) is an agonist of δ-opioid receptor.
-
In Vitro——
-
In VivoTwice daily administration of Deltorphin I (20μg/mouse) for 4 days produces tolerance to Deltorphin I analgesia, as shown by the decrease in the analgesic response. The peak analgesic response to Deltorphin I (20 μg/mouse) at 10 min after injections is decreased from 8.36±0.28 s (the 1st day) to 4.53±0.14 s (the 4th day) markedly. Concurrent treatment of Melatonin (0.5, 1 and 2.5 mg/kg) and Deltorphin I (20 μg/mouse) twice daily for 4 days can attenuate the tolerance to Deltorphin I analgesia (P<0.05, <0.05 and <0.05), and this effect is dose dependent.
-
SynonymsDeltorphin 1 | Deltorphin C
-
PathwayEndocrinology/Hormones
-
TargetOpioid Receptor
-
Recptorδ-opioid receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number122752-15-2
-
Formula Weight768.86
-
Molecular FormulaC37H52N8O10
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 25 mg/mL (32.52 mM)
-
SMILESCC(C)[C@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@H](C(=O)NCC(N)=O)C(C)C
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Dupin S Tafani J A M Honoré Mazarguil et al. [125I][D-Ala2]deltorphin-I: A high affinity delta-selective opioid receptor ligand[J]. Peptides 1991 12(4):825-830.
molnova catalog
related products
-
Deltorphin 2(TFA)
Deltorphin 2(TFA) is an agonist of δ opioid receptor(IC50:0.41 nM).
-
Ac-RYYRIK-NH2
High affinity ligand for the NOP site (Ki = 1.5 nM). Antagonizes nociceptin-stimulated GTP binding in rat brain and the chronotropic effect of nociceptin on rat cardiomyocytes. However, displays potent agonist properties in vivo, inhibiting locomotor activity in mice.
-
Adrenorphin 3TFA(883...
Adrenorphin(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
